Kinase test results (IC50 values in micromoles) from the manuscript Jorda et al. - "How selective are pharmacological inhibitors of cyclin-dependent kinases?" (submitted):
heatcolours: IC50 heat colours: IC50 for each inhibitor scaled to [0,1]) heat colours: logIC50 for each inhibitor scaled to [0,1])

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	CDK1/B	CDK2/E	CDK2/A	CDK4/D1	CDK5/p25	CDK7/H	CDK9/T
Dinaciclib	0.072	0.0034	0.0039	0.11	0.045	0.17	0.18
R-CR8	0.79	0.036	0.14	10	0.68	1.8	0.99
JNJ7706621	0.02	0.0018	0.0018	0.56	0.017	1.2	0.061
SNS032	0.2	0.0045	0.023	0.45	0.44	0.29	0.048
Flavopiridol	0.49	0.23	0.084	0.21	0.26	0.82	0.025
CDK2/9 inhibitor	0.15	0.01	0.01	0.66	0.19	0.17	0.051
BML259	1.7	0.2	0.35	10	0.46	0.64	3.4
BIO	0.27	0.014	0.069	0.53	0.041	3.5	0.45
PNU112455A	5.3	1.9	0.95	10	4.4	10	10
(R)-DRF053	3.7	0.093	0.29	10	0.21	0.82	8
CDK1/5 inhibitor	9.7	5.6	4.4	10	10	10	10
CDK1/2 inhibitor III	0.0021	0.0028	0.0002	0.059	0.0002	0.066	0.03
BMS265246	0.014	0.0056	0.071	0.22	0.26	1.6	1.8
NU6102	0.15	0.022	0.014	0.18	0.12	2.5	4.1
CGP60474	0.026	0.003	0.0041	0.22	0.0095	0.2	0.013
CDK9-IN-2	0.55	0.15	0.17	1.8	1.1	2.3	0.033
LDC000067	4	2.3	1.1	3.2	5	10	0.23
CDK-IN-2	0.22	0.86	0.32	0.63	7.3	4.9	0.05
PHA767491	1.1	1.2	0.64	10	1	10	0.076
BS181	10	1.4	1.3	10	4.3	0.11	1.8
Ribociclib	10	10	10	0.03	10	10	3.9
ON123300	0.6	0.38	0.055	0.018	0.27	6	0.12
Abemaciclib	0.37	0.35	0.046	0.0052	0.4	3.1	0.1
CDK4 inhibitor V	0.29	0.5	0.071	0.038	1.2	10	1
Palbociclib	9.8	9.1	1.8	0.013	10	10	1.1
CDK4 inhibitor	1.5	0.23	0.19	0.091	0.15	10	4
Arcyriaflavin A	0.96	0.53	0.14	3.1	0.94	10	10
CINK4	9.2	5.2	10	10	10	10	10
Ryuvidine	10	10	10	9.5	10	10	10
NSC625987	10	10	10	10	10	10	10
Milciclib	1.2	0.59	0.11	0.22	0.38	0.27	7.7
NU6140	5.5	1.2	0.41	0.94	8.8	2.3	5.1
SU9516	0.17	0.026	0.027	1.7	0.022	0.9	1.5
CDK2 inhibitor II	1.3	0.031	0.041	2.8	0.74	10	1.1
GW8510	0.049	0.0028	0.0033	0.14	0.0067	0.32	0.54
CVT313	3.7	0.18	0.22	10	0.42	9.2	2.3
RO3306	0.047	0.19	0.25	10	2.5	10	10
Elbfluorene	10	10	10	10	10	10	10
Benfluorene	10	10	7.1	10	10	10	10
CDK1 inhibitor	6.7	9.4	10	10	5.8	10	10
CGP74514A	0.15	0.026	0.046	3	0.026	0.28	1.4

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